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Pasireotide (diaspartate)

CAT: 0931-T75248-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T75248-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1421446-02-7
Target
Others, Somatostatin
Related Pathways
GPCR/G Protein, Others
Bioactivity
Pasireotide diaspartate (SOM230), a long-acting cyclohexapeptide and somatostatin analog, enhances agonist activity across somatostatin receptor subtypes (sst1/2/3/4/5, with pK i values of 8.2, 9.0, 9.1, <7.0, and 9.9, respectively) . This compound demonstrates antisecretory, antiproliferative, and proapoptotic activities [1] [2].
Smiles
OC(C[C@H](N)C(O)=O)=O.O=C1N2[C@@](C(N[C@@H](C3=CC=CC=C3)C(N[C@@H](C(N[C@H](C(N[C@H](C(N[C@H]1CC4=CC=CC=C4)=O)CC5=CC=C(C=C5)OCC6=CC=CC=C6)=O)CCCCN)=O)CC7=CNC8=CC=CC=C78)=O)=O)([H])C[C@H](C2)OC(NCCN)=O.OC(C[C@H](N)C(O)=O)=O
Molecular Formula
C66H80N12O17
Molecular Weight
1313.41
Shipping Conditions
Ice Packs
Storage Temperature
-20°C