Pasireotide

• Target:

  Somatostatin|||Others

• Related Pathways:

  GPCR/G Protein|||Others

• Bioactivity:

  Pasireotide (SOM 230) is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9 respectively) .

• Smiles:

  O=C1N2[C@@](C[C@@H](OC(NCCN)=O)C2)(C(=O)N[C@](C(=O)N[C@H](CC=3C=4C(NC3)=CC=CC4)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC5=CC=C(OCC6=CC=CC=C6)C=C5)C(=O)N[C@H]1CC7=CC=CC=C7)(C8=CC=CC=C8)[H])[H]

• Molecular Formula:

  C58H66N10O9

• Molecular Weight:

  1047.21

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  396091-73-9