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JHDM-IN-1

CAT: 0931-T75175-01Size: 100 mgDry Ice: NoHazardous: No
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CAT#:0931-T75175-01Size:100 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1310809-17-6
Target
Others, Histone Demethylase
Related Pathways
Others, Chromatin/Epigenetic
Bioactivity
JHDM-IN-1 (Compound 1), a Jumonji C domain-containing HDMs (JHDM) inhibitor, exhibits IC50s of 3.4 μM against JMJD2C, 4.3 μM against JMJD2A, 5.9 μM against JMJD2E, 10 μM against PHF8, and 43 μM against JMJD3, showcasing its inhibitory effectiveness across a spectrum of JHDM enzymes [1].
Smiles
N(C(OCC1=CC=C(CNCCCCN(C(/C=C/C(O)=O)=O)O)C=C1)=O)C=2C3=C(C=CC2)C=CC=C3
Molecular Formula
C27H29N3O6
Molecular Weight
491.54
Shipping Conditions
Ice Packs
Storage Temperature
-20°C