Bromodomain IN-2

CAT: 0931-MF-0154986-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0154986-01Size:5 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2445335-77-1
Target
Epigenetic Reader Domain|||Others
Related Pathways
Chromatin/Epigenetic|||Others
Bioactivity
BD-IN-1, a pan bromodomain (BD) inhibitor, exhibits K_D values of 250 nM for BRD4 (1), 420 nM for CBP, 130 nM for BRPF1B, 430 nM for BRD7, 67 nM for BRD9, 240 nM for BRDT (1), and 970 nM for CECR2, respectively. This compound demonstrates antiproliferative activity [1].
Smiles
ClC1=C(C2=C3C(=C(C)N2)C(=O)CCCC3)C=C(N)C=C1
Molecular Formula
C16H17ClN2O
Molecular Weight
288.77
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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