GCGR antagonist 2

CAT: 0931-T72621-01Size: 25 mgDry Ice: NoHazardous: No

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CAT#:0931-T72621-01Size:25 mg

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24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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CAS Number

280134-25-0

Target

Glucagon Receptor, Others

Related Pathways

Others, GPCR/G Protein

Bioactivity

GCGR Antagonist 2, a Furan-2-carbohydrazide, serves as an orally active antagonist of the glucagon receptor. It exhibits affinity for the human glucagon receptor (hGluR) with a dissociation constant (Kd) of 2.3 nM and demonstrates inhibitory activity against the rat receptor with a half-maximal inhibitory concentration (IC50) of 0.43 nM. Additionally, this compound effectively prevents glucagon-stimulated glycogenolysis.

Smiles

C(N1C=2C(=C(C=NNC(=O)C3=CC(C#N)=C(O)C=C3)C=CC2)C=C1)C4=C(C)C(C)=CC(C)=C4C

Molecular Formula

C28H26N4O2

Molecular Weight

450.53

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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