YM-58790

• Target:

  AChR

• Related Pathways:

  Neuroscience

• Purity:

  0.9987

• Bioactivity:

  YM-58790 free base is a potent mAChR antagonist that inhibits M1 mAChR, M2 mAChR, and M3 mAChR with Ki values of 28 nM, 260 nM, and 15 nM, respectively. It inhibits reflex rhythmic bladder contractions in rats by inhibiting bladder pressurization.

• Smiles:

  C(NC(OC1CCN(CC2=CC=C(NC)C=C2)CC1)=O)(C3=CC=CC=C3)C4=CC=CC=C4

• Molecular Formula:

  C27H31N3O2

• Molecular Weight:

  429.55

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  168830-70-4