TRPM8 antagonist 4

CAT: 0931-T211390-01Size: 10 mgDry Ice: NoHazardous: No

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CAT#:0931-T211390-01Size:10 mg

Selected

24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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Target

Interleukin, Cannabinoid Receptor, TRP/TRPV Channel, TNF

Related Pathways

GPCR/G Protein, Apoptosis, Immunology/Inflammation, Membrane transporter/Ion channel

Bioactivity

TRPM8 antagonist 4 is a compound with high functional selectivity and favorable physicochemical properties, serving as a CB2R partial agonist (EC50=54.2 μM, Ki=3.2 μM) and a TRPM8 (IC50=42.3 nM) antagonist. It possesses notable anti-inflammatory and analgesic effects, demonstrating good safety by reducing the mRNA expression of TNF-α, IL-6, and IL-1β.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

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HY-112430-01	TRPM8 antagonist 2
M28848-01	TRPM8 antagonist 3
GTR19263785-01	TRPM8 antagonist 4
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A19329-1	TRPM8 antagonist 2 1mg
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A19329-100	TRPM8 antagonist 2 100mg
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TRPM8 antagonist 4

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