Products for Research Use Only

ENX-101

CAT: 0931-T206766-01Size: 10 mgDry Ice: NoHazardous: No
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CAT#:0931-T206766-01Size:10 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
GABA Receptor
Related Pathways
Neuroscience, Membrane transporter/Ion channel
Bioactivity
ENX-101 is an orally active partial positive allosteric modulator (PAM) of the (GABAA) receptor. It selectively targets the α2β2γ2L (EC50= 0.76 nM), α2β3γ2L (EC50= 0.61 nM), α3 (EC50= 1.97 nM), and α5 (EC50= 0.85 nM) subunits of the GABA receptor. ENX-101 demonstrates anticonvulsant activity in various animal models.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C