RTI-122

• Target :

  GPCR

• Related Pathways :

  GPCR/G Protein|||Endocrinology/Hormones

• Bioactivity :

  RTI-122 is an effective GPR88 agonist with good metabolic stability (half-life of 5.8 hours in mice) and a cAMP EC50 of 11 nM. It can penetrate the blood-brain barrier and is utilized in research related to excessive drinking.

• Smiles :

  C(N(C[C@H]([C@H](OC)C)N)C1=CC=C(C=C1)C2=CC=C(OC(C)C)C=C2)(=O)[C@H]3[C@@H](C3)C4=CC=C(F)C=N4

• Molecular Formula :

  C29H34FN3O3

• Molecular Weight :

  491.6

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  3034664-39-3