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GA-017

CAT: 0957-E1145-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0957-E1145-01Size:5 mg
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Description
GA-017 inhibits the serine/threonine protein kinases large tumor suppressor kinase 1/2 (LATS1/2), which exerts inhibitory with IC50s against LATS1 and 2 of 4.10±0.79 and 3.92±0.42 nM, respectively, and competitively inhibits LATS1 and 2 against ATP, with Ki (inhibition constant) values of 0.58±0.11 and 0.25±0.03 nM, respectively.
CAS Number
2351906-74-4
Target
LATS
Activity
Hippo
Molecular Formula
C18H21N3O4
Storage Conditions
3 years -20°C powder