ABX-1431

CAT: 0498-bs-82936C-01Size: 10 mgDry Ice: NoHazardous: No
CAT#: bs-82936C-01Size: 10 mg
Selected
AVAILABILITY
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Background
Potent (IC50 = 14 nM in vitro, 2.2 nM in human PC3 cells) and very selective (>100-fold over hABHD6, >200-fold over hPLA2G7) inhibitor of monoacylglycerol lipase (MAGL) .1 Active in a rat formalin pain test at 3mg/kg. Orally bioavailable and CNS penetrant.
Conjugation
Unconjugated
Buffer
White solid
Storage Conditions
-20°C