GSK-J1

CAT: 0498-bs-82218C-01Size: 5 mgDry Ice: NoHazardous: No

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CAT#:0498-bs-82218C-01Size:5 mg

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24/48H Stock Items & 2 to 6 Weeks non Stock Items.

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Background

Potent and selective inhibitor of jumonji H3K27 histone demethylases JMJD3 and UTX (IC50 = 60 nM, human JMJD3) . This is the first known inhibitor selective for the H3K27me3-specific JMJ subfamily which binds to the active catalytic site of the enzyme. The COOH group confers cell impermeability and as such is useful as a standard in in vitro assays. A cell permeable ethyl ester analog is also available.

Conjugation

Unconjugated

Buffer

Pale yellow solid

Storage Conditions

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HY-15648-01	GSK-J1
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GSK-J1

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