UFP-101

• Description:

  Potent, selective and competitive silent antagonist for the NOP opioid receptor. Binds to NOP with high affinity (pKi = 10.24) and displays > 3000-fold selectivity over δ, μ and κ opioid receptors. Antinociceptive and opposes the action of nociceptin in vivo.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  1908.19

• Molecular Formula:

  C82H138N32O21

• Notes:

  Research use only, not for human use.

• Receptor:

  ——

• CAS Number:

  849024-68-6