CB2R PAM

• Description:

  CB2R PAM is an orally active cannabinoid type 2 receptor (CB2Rs) positive allosteric modulator that enhances CP 55940 and 2-Arachidonylglycerol-stimulated [35S]GTPγS binding to CB2 receptors without affecting receptor activity in the absence of agonists. CB2R PAM shows anti-injury activity in a mouse model of neuropathic pain.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  435.33

• Molecular Formula:

  C21H24BrFN2O2

• Notes:

  Research use only, not for human use.

• Receptor:

  Cannabinoid Receptor

• CAS Number:

  2244579-87-9