BRD7-IN-1

• Description :

  BRD7-IN-1, a modified derivative of BI7273 (BRD7/9 inhibitor), forms PROTAC VZ185 via linkage to a VHL ligand, demonstrating potent activity against BRD7/9 with DC50 values of 4.5 and 1.8 nM, respectively .

• Stability :

  ≥ 2 years

• Purity :

  >98% (HPLC)

• Weight :

  467.39

• Molecular Formula :

  C22H28Cl2N4O3

• Notes :

  Research use only, not for human use.

• Receptor :

  Epigenetic Reader Domain

• CAS Number :

  2448414-48-8