BRD7-IN-1

• Description:

  BRD7-IN-1, a modified derivative of BI7273 (BRD7/9 inhibitor), forms PROTAC VZ185 via linkage to a VHL ligand, demonstrating potent activity against BRD7/9 with DC50 values of 4.5 and 1.8 nM, respectively .

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  467.39

• Molecular Formula:

  C22H28Cl2N4O3

• Notes:

  Research use only, not for human use.

• Receptor:

  Epigenetic Reader Domain

• CAS Number:

  2448414-48-8