MK-6892

• Description:

  MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: 4 nM; GTPγS EC50: 16 nM) .MK-6892 evokes a potent internalization of GPR109A in U2OS β-arrestin2-RrGFP cells.MK-6892 shows an EC50 value of 74 nM on calcium mobilization assay.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  386.4

• Molecular Formula:

  C19H22N4O5

• Notes:

  Research use only, not for human use.

• Receptor:

  GPR109A

• CAS Number:

  917910-45-3