THZ 531

• Description:

  THZ 531 (THZ531) is a first-in-class, selective CDK12 and CDK13 covalent inhibitor with IC50 of 158 nM and 69 nM, respectively.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  558.083

• Molecular Formula:

  C30H32ClN7O2

• Notes:

  Research use only, not for human use.

• Receptor:

  CDK12, CDK13

• CAS Number:

  1702809-17-3