BS-194

• Description:

  BS-194 is a potent, selective, orally bioactive CDK2 inhibitor with IC50 of 2.4 nM, displays 140-fold selectivity over CDK7 (IC50=378 nM) ; weakly inhibits CDK1, CDK5, CDK7, and CDK9 with IC50 of 30, 30, 250, and 90 nM.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  385.468

• Molecular Formula:

  C20H27N5O3

• Notes:

  Research use only, not for human use.

• Receptor:

  CDK

• CAS Number:

  1092443-55-4