RVX-208

• Description:

  RVX-208 is a potent BET bromodomain inhibitor with IC50 of 0.510 μM for BD2 in a cell-free assay, about 170-fold selectivity over BD1. Phase 2.

• Stability:

  ≥ 2 years

• Purity:

  >98% (HPLC)

• Weight:

  370.4

• Molecular Formula:

  C20H22N2O5

• Notes:

  Research use only, not for human use.

• Receptor:

  BD2

• CAS Number:

  1044870-39-4