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Apabetalone (RVX-208)

CAT: 0957-S7295-01Size: 5 mgDry Ice: YesHazardous: No
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CAT#:0957-S7295-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Apabetalone (RVX-208, RVX-000222) is a potent BET bromodomain inhibitor with IC50 of 0.510 μM for BD2 in a cell-free assay, about 170-fold selectivity over BD1. Phase 2.
CAS Number
1044870-39-4
Synonyms
RVX-000222
Target
Epigenetic Reader Domain
Activity
Epigenetics
Molecular Formula
C20H22N2O5
Storage Conditions
2 years -80 in solvent