(2R,3R) -E1R

CAT: 0804-HY-116463C-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0804-HY-116463C-01Size:5 mg
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
Description
(2R,3R) -E1R (Compound 2b) is an enantiomer of E1R. (2R,3R) -E1R is a sigma-1 receptor positive allosteric modulator (Sig1R PAM) for the treatment of cognition/memory disorders[1].
CAS Number
[1400888-63-2]
UNSPSC
12352005
Target
Sigma Receptor
Type
Reference compound
Related Pathways
Neuronal Signaling
Applications
Neuroscience-Neurodegeneration
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/2r-3r-e1r.html
Purity
98.79
Solubility
DMSO : 50 mg/mL (ultrasonic)
Smiles
O=C(N)CN1[C@H](C)[C@@H](C2=CC=CC=C2)CC1=O
Molecular Formula
C13H16N2O2
Molecular Weight
232.28
References & Citations
[1]Veinberg G, et al. Synthesis and biological evaluation of 2- (5-methyl-4-phenyl-2-oxopyrrolidin-1-yl) -acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor. Bioorg Med Chem. 2013 May 15;21 (10) :2764-71.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
Sigma 1 Receptor

Related Products

CatalogName
HY-116463A-01(2R,3S) -E1R
HY-N13500(2R,3R) -Glucodistylin
HY-138563A-01(2R,3R) -GSK973
HY-137440B-01(2R,3R) -Firazorexton
HY-116463-01E1R
HY-122311ABis (2R,3R) -Orniplabin
HY-B0632B(2R,3R) -Diltiazem (hydrochloride)
HY-116463D-01(Rac) -E1R
HY-78932D(2R,3R) -Dap-NE (hydrochloride)
HY-116463B-01(2S,3S) -E1R

Alternative Products

CatalogName
MBS5752603(2R,3R)-E1R
MF-0002636-01(2R,3R) -E1R
MBS5752605(2R,3S)-E1R
MF-0002643-01(2R,3S) -E1R
MF-0004158-01E1R
018634(2R,3R,4R) -
MF-0002637(2R,3R) -Glucodistylin
MBS6072351-01(2R,3R,4R)-
MBS5788360(2R,3R)-Glucodistylin
MBS3609571-01(2R, 3R)-(-)-23-Butanediol

Popular Products