IPR-803

CAT: 0804-HY-111192-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0804-HY-111192-01Size:5 mg
Selected
PRICE
AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Product image 1
1 / 1
Description
IPR-803 is a potent inhibitor of the uPARĀ·uPA protein-protein interaction (PPI) . IPR-803 binds directly to uPAR with sub-micromolar affinity. IPR-803 displays anti-tumor activity[1].
CAS Number
[892243-35-5]
UNSPSC
12352005
Target
Ser/Thr Protease
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ipr-803.html
Purity
98.0
Solubility
DMSO : 7.69 mg/mL (ultrasonic)
Smiles
O=C(O)C1=CC=CC(NC2=C(C3=C4ON=C3C(N5CCCCCC5)=C2)C(C6=C4C=CC=C6)=O)=C1
Molecular Formula
C27H23N3O4
Molecular Weight
453.49
References & Citations
[1]Mani T, et al. Small-molecule inhibition of the uPARā€¢uPA interaction: synthesis, biochemical, cellular, in vivo pharmacokinetics and efficacy studies in breast cancer metastasis. Bioorg Med Chem. 2013 Apr 1;21 (7) :2145-55.
Shipping Conditions
Room Temperature
Storage Conditions
-20Ā°C, 3 years; 4Ā°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

Related Products

CatalogName
HY-P1166UFP-803
HY-W999618CRBN ligand-803
HY-10780JTV-803 (mesylate)
HY-P1166AUFP-803 (TFA)
HY-W043473-01Fmoc-Lys (ipr, Boc) -OH
HY-13299-01MK-8033
HY-149051-01BGB-8035
HY-107143BL-8030
HY-167894DA-8031
HY-13299A-01MK-8033 (hydrochloride)

Alternative Products

CatalogName
MBS3614899-01IPR-803
MBS5774575SRPIN-803
MF-0109903UFP-803
66068-84-6Sandenol 803
MBS5764097UFP 803
MBS5784812ZYZ-803
MBS9022817-01Fmoc-Ser(iPr)-OH
5-05909Boc-Lys(iPr)-OH
5-06698Fmoc-Lys(ipr)-OH
BLG-I0072ā€²,3ā€²-Ipr-Guo

Popular Products