Products for Research Use Only

D3R/MOR antagonist 1

CAT: 0013-GTR19230933-01Size: 50 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19230933-01Size:50 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Compound 114 is a dual D3 dopamine and mu-opioid receptor antagonist with K i values of 46.5 nM and 691 nM, respectively. Its MOR partial agonism provides analgesic potential, while D3R antagonism may mitigate abuse liability, supporting research in neuropharmacology and addiction studies.
Field of Research
Metabolism Research, Neuroscience, Neuroscience; Pharmacology & Drug Discovery, Pharmacology & Drug Discovery
Molecular Formula
C22H27Cl2N3O
Molecular Weight
420.38
Storage Conditions
-20°C
Notes
For research use only.