Products for Research Use Only

D3R/MOR antagonist 2

CAT: 0013-GTR19230932-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19230932-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
Compound 121 is a dual D3 receptor antagonist (K i = 361 nM) and mu-opioid receptor antagonist/partial agonist (K i = 85.2 nM) . This profile suggests utility in preclinical research for investigating novel analgesic mechanisms with potentially reduced abuse liability, applicable in both in vitro binding assays and in vivo behavioral models.
Field of Research
Metabolism Research, Neuroscience, Neuroscience; Pharmacology & Drug Discovery, Pharmacology & Drug Discovery
Molecular Formula
C25H31ClN2O
Molecular Weight
410.98
Storage Conditions
-20°C
Notes
For research use only.