Products for Research Use Only

PDE1-IN-5

CAT: 0013-GTR19230846-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19230846-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PDE1-IN-5 (Compound 10c) is a potent and selective PDE1C inhibitor (IC50 = 15 nM) with demonstrated anti-inflammatory activity. It suppresses LPS-induced pro-inflammatory mediators like iNOS, TNF-α, and interleukins. Its efficacy in reducing colitis symptoms in a DSS-induced mouse model highlights its utility for inflammatory disease research, particularly for studying IBD mechanisms.
Field of Research
Metabolism Research
Molecular Formula
C27H29FN4O
Molecular Weight
444.54
Storage Conditions
-20°C
Notes
For research use only.