Products for Research Use Only

RORγ antagonist 1

CAT: 0013-GTR19230521-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19230521-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
RORγ antagonist 1 is a potent betulinic acid derivative functioning as a RORγ antagonist (K D = 0.18 μM) . It exhibits anti-proliferative activity in pancreatic cancer models, suppressing RAS/MAPK and AKT/mTORC1 pathways while inducing caspase-dependent apoptosis in vitro and in vivo.
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Molecular Formula
C35H60N2O2
Molecular Weight
540.86
Storage Conditions
-20°C
Notes
For research use only.