Products for Research Use Only

GB-88

CAT: 0013-GTR19205811Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19205811Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
GB-88 is a selective, orally bioavailable non-peptide antagonist of protease-activated receptor 2 (PAR2) . It inhibits PAR2-mediated calcium mobilization with an IC50 of 2 μM, making it a useful tool for investigating PAR2's role in inflammation and pain in both cellular and animal models.
CAS Number
1416435-96-5
Field of Research
Pharmacology & Drug Discovery
Smiles
C ([C@@H] (NC ([C@H] (CC1CCCCC1) NC (=O) C2=CC=NO2) =O) [C@H] (CC) C) (=O) N3CCC4 (C=5C (C=C4) =CC=CC5) CC3
Molecular Formula
C32H42N4O4
Molecular Weight
546.70
Storage Conditions
-20°C
Notes
For research use only.

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