Products for Research Use Only

LX-039

CAT: 0013-GTR19185497-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19185497-01Size:25 mg
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Description
LX-039 is a potent and selective oral estrogen receptor degrader (SERD) with an EC50 of 2.99 nM, featuring an indole C-3 chloride substitution. It demonstrates favorable pharmacokinetics with low clearance and high oral exposure in mice, supporting its investigation for antitumor efficacy in breast cancer research models.
CAS Number
2135341-09-0
Field of Research
Metabolism Research
Smiles
C (=C (CC) C1=C (Cl) C=C (F) C=C1) (C2=C (Cl) C=3C (N2) =CC=CC3) C4=CC=C (C=CC (O) =O) C=C4
Molecular Formula
C27H20Cl2FNO2
Molecular Weight
480.36
Storage Conditions
-20°C
Notes
For research use only.