Products for Research Use Only

BRD4 Inhibitor-10

CAT: 0013-GTR19175096-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19175096-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
BRD4 Inhibitor-10 is a potent and selective small molecule targeting the first bromodomain (BD1) of BRD4 with an IC50 of 8 nM. This compound is a valuable chemical probe for epigenetic research, utilized in vitro to study transcriptional regulation in oncology and inflammation, and has been employed in vivo in preclinical cancer models.
CAS Number
1660117-38-3
Product Name Alternative
BRD4-BD1, BRD4 Inhibitor 10, BRD4 Inhibitor10, BRD-4 Inhibitor-10, BRD4 Inhibitor-10, inhibit, Inhibitor, EpigeneticReaderDomain, Epigenetic Reader Domain
Field of Research
Epigenetics & Chromatin, Epigenetics & Chromatin; Pharmacology & Drug Discovery
Purity
98.98% (May vary between batches)
Solubility
DMSO:125 mg/mL (291.03 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (9.31 mM)
Smiles
C[C@@H] (c1ccccc1) n1c (nc2cnc (cc12) C1CCOCC1) -c1cc (C) c (=O) n (C) n1
Molecular Formula
C25H27N5O2
Molecular Weight
429.51
Storage Conditions
-20°C
Notes
For research use only.