Products for Research Use Only

GSK046

CAT: 0013-GTR19167001-01Size: 1 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0013-GTR19167001-01Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Description
GSK046 (iBET-BD2) is a selective, orally bioavailable inhibitor targeting the second bromodomain (BD2) of BET proteins, exhibiting potent immunomodulatory activity. It is widely used in research to investigate BET protein function in inflammatory and oncological contexts, with applications in both cellular assays and in vivo models.
CAS Number
2474876-09-8
Product Name Alternative
GSK046, GSK-046, GSK 046, Epigenetic Reader Domain, EpigeneticReaderDomain, iBET-BD2, Inhibitor, immuno-inflammation, inhibit, BD2, BRD2-BD2, BRD2, BRD3-BD2, BRD3, BRD4, BRDT-BD2, BRDT, BRD4-BD2
Field of Research
Epigenetics & Chromatin
Purity
99.94% (May vary between batches)
Solubility
DMSO:83.33 mg/mL (201.05 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:3.3 mg/mL (7.96 mM)
Smiles
C[C@H] (Oc1cc (cc (F) c1NC (C) =O) C (=O) N[C@H]1CC[C@H] (O) CC1) c1ccccc1
Molecular Formula
C23H27FN2O4
Molecular Weight
414.47
Storage Conditions
-20°C
Notes
For research use only.