Products for Research Use Only

PEN-221

CAT: 0013-GTR19036844-01Size: 100 mgDry Ice: NoHazardous: No
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CAT#:0013-GTR19036844-01Size:100 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
PEN-221 is a cytotoxic drug conjugate that selectively targets the somatostatin receptor subtype 2 (SSTR2) with an IC50 of 10 nM. It consists of the microtubule-disrupting agent DM1 conjugated to Tyr3-octreotate, enabling targeted delivery to SSTR2-expressing cells. This construct is used in preclinical research for investigating targeted cancer therapies, including in vitro cytotoxicity assays and in vivo xenograft models for neuroendocrine and other SSTR2-positive tumors.
Molecular Weight
1786.55
Storage Conditions
-20°C
Notes
For research use only.