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(R) -PS210

CAT: 0804-HY-13856-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0804-HY-13856-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Description
(R) -PS210, the R enantiomer of PS210 (compound 4h-eutomer), is a substrate-selective allosteric activator of PDK1 with an AC50 value of 1.8 μM. (R) -PS210 targets to the PIF-binding pocket of PDK1. PIF: The protein kinase C-related kinase 2 (PRK2) -interacting fragment[1].
CAS Number
1410101-89-1
UNSPSC
12352005
Target
PDK-1
Type
Reference compound
Related Pathways
PI3K/Akt/mTOR
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/r-ps210.html
Purity
98.09
Solubility
DMSO : 230 mg/mL (ultrasonic)
Smiles
O=C(O)C([C@H](C1=CC=CC=C1)CC(C2=CC=C(C(F)(F)F)C=C2)=O)C(O)=O
Molecular Formula
C19H15F3O5
Molecular Weight
380.31
References & Citations
[1]Wilhelm A, et al. 2- (3-Oxo-1,3-diphenylpropyl) malonic acids as potent allosteric ligands of the PIF pocket of phosphoinositide-dependent kinase-1: development and prodrug concept.J Med Chem. 2012 Nov 26;55 (22) :9817-30.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported

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