STAT5-IN-2
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


STAT5-IN-2
UNSPSC Description:
STAT5-IN-2 is a STAT5 inhibitor, extracted from reference 1, example 17f. STAT5-IN-2 has potent antileukemic effect[1].Target Antigen:
Apoptosis; STATType:
Reference compoundRelated Pathways:
Apoptosis;JAK/STAT Signaling;Stem Cell/WntApplications:
Cancer-Kinase/proteaseField of Research:
CancerAssay Protocol:
https://www.medchemexpress.com/STAT5-IN-2.htmlPurity:
99.08Solubility:
DMSO : 100 mg/mL (ultrasonic)Smiles:
CC(CCN1CCOC2=CC(C=CN3)=C3C=C2)(C)C4=C1C=CC(C5=CC=CN=C5)=C4Molecular Weight:
397.51References & Citations:
[1]Ludovic Juen, et al. New Inhibitor Targeting Signal Transducer and Activator of Transcription 5 (STAT5) Signaling in Myeloid Leukemias. J Med Chem. 2017 Jul 27;60(14):6119-6136.Shipping Conditions:
Room TemperatureStorage Conditions:
-20°C, 3 years; 4°C, 2 years (Powder)Clinical Information:
No Development ReportedCAS Number:
2111834-61-6
