NI-57
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


NI-57
Target:
Epigenetic Reader DomainRelated Pathways:
Chromatin/EpigeneticPurity:
>99.99%Bioactivity:
NI-57 is an inhibitor of the bromodomain and plant homeodomain finger-containing (BRPF) family proteins, with IC50 values of 3.1 nM for BRPF1, 46 nM for BRPF2 (BRD1), and 140 nM for BRPF3.Smiles:
COc1cc (ccc1S (=O) (=O) Nc1ccc2n (C) c (=O) c (C) cc2c1) C#NMolecular Formula:
C19H17N3O4SMolecular Weight:
383.42Shipping Conditions:
Cool packStorage Temperature:
-20°CCAS Number:
1883548-89-7
