NI-57
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


NI-57
Target :
Epigenetic Reader DomainRelated Pathways :
Chromatin/EpigeneticPurity :
>99.99%Bioactivity :
NI-57 is an inhibitor of the bromodomain and plant homeodomain finger-containing (BRPF) family proteins, with IC50 values of 3.1 nM for BRPF1, 46 nM for BRPF2 (BRD1), and 140 nM for BRPF3.Smiles :
COc1cc(ccc1S(=O)(=O)Nc1ccc2n(C)c(=O)c(C)cc2c1)C#NMolecular Formula :
C19H17N3O4SMolecular Weight :
383.42Shipping Conditions :
Cool packStorage Temperature :
-20°CCAS Number :
1883548-89-7

