MI-503
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


MI-503
Target :
Histone Methyltransferase|||Epigenetic Reader DomainRelated Pathways :
Chromatin/EpigeneticPurity :
0.9999Bioactivity :
MI-503 is an efficient and selective Menin-MLL inhibitor with an IC50 of 14.7 nM. In human MLL leukemia cell lines, MI-503 has a significant growth inhibition effect (GI = 250 nM-570 nM) .Smiles :
Cc1c(CN2CCC(CC2)Nc2ncnc3sc(CC(F)(F)F)cc23)ccc2n(Cc3cn[nH]c3)c(cc12)C#NMolecular Formula :
C28H27F3N8SMolecular Weight :
564.63Shipping Conditions :
Cool packStorage Temperature :
-20°CCAS Number :
1857417-13-0

