CCG-273463

• Target:

  Others|||GRK

• Related Pathways:

  GPCR/G Protein|||Others

• Bioactivity:

  CCG-273463 is a potent, covalent, selective inhibitor of GRK5 (IC50: 9 nM) . CCG-273463 can be used to study heart failure, hypertrophic cardiomyopathy and cancer.

• Smiles:

  C (=C\1/C=2C (NC1=O) =CC=C (C (N[C@H] (C) C3=CC=CC=C3) =O) C2) \C4=C (C) C (NC (CBr) =O) =C (C) N4

• Molecular Formula:

  C26H25BrN4O3

• Molecular Weight:

  521.41

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2750413-99-9