CCG-273463

• Target :

  Others|||GRK

• Related Pathways :

  GPCR/G Protein|||Others

• Bioactivity :

  CCG-273463 is a potent, covalent, selective inhibitor of GRK5 (IC50: 9 nM) . CCG-273463 can be used to study heart failure, hypertrophic cardiomyopathy and cancer.

• Smiles :

  C(=C\1/C=2C(NC1=O)=CC=C(C(N[C@H](C)C3=CC=CC=C3)=O)C2)\C4=C(C)C(NC(CBr)=O)=C(C)N4

• Molecular Formula :

  C26H25BrN4O3

• Molecular Weight :

  521.41

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2750413-99-9