GRK5-IN-3

• Target :

  Others|||GRK

• Related Pathways :

  Others|||GPCR/G Protein

• Bioactivity :

  GRK5-IN-3 is a covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5), significantly inhibiting GRK5 with an IC50 of 0.22 ?M and GRK6 with an IC50 of 0.41 ?M.

• Smiles :

  N(C1=C2C(=NC(NC3=C(OC)C=C(NC(C=C)=O)C=C3)=N1)NC=C2)C4=C(C(N)=O)C=CC=C4

• Molecular Formula :

  C23H21N7O3

• Molecular Weight :

  443.46

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2410793-22-3