GRK5-IN-4

• Target :

  Others|||GRK

• Related Pathways :

  GPCR/G Protein|||Others

• Bioactivity :

  GRK5-IN-4 is a selective, potent, covalent GRK5 (G protein-coupled receptor kinase 5) inhibitor (IC50: 1.1 ?M) .GRK5-IN-4 is 90 times more selective for GRK5 than GRK2.GRK5-IN-4 can be used to study heart failure.

• Smiles :

  N(C1=C2C(=NC(NC3=C(OC)C=C(CNC(C#CC)=O)C=C3)=N1)NC=C2)C4=C(C(NC)=O)C=CC=C4

• Molecular Formula :

  C26H25N7O3

• Molecular Weight :

  483.52

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2410794-89-5