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PFI-1

CAT: 0931-T6222-01Size: 5 mgDry Ice: NoHazardous: No
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CAT#:0931-T6222-01Size:5 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1403764-72-6
Target
Epigenetic Reader Domain, Apoptosis, Autophagy
Related Pathways
Chromatin/Epigenetic, Apoptosis, Autophagy
Purity
0.9919
Bioactivity
PFI-1 (PF-6405761), a specific BET (bromodomain-containing protein) inhibitor for BRD4, is with the IC50 of 0.22 μM in a cell-free assay.
Smiles
COc1ccccc1S(=O)(=O)Nc1ccc2NC(=O)N(C)Cc2c1
Molecular Formula
C16H17N3O4S
Molecular Weight
347.39
Shipping Conditions
Ice Packs
Storage Temperature
-20°C