PFI-1

CAT:
931-T6222-01
Size:
5 mg
  • Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
  • Dry Ice Shipment: No
PFI-1 - image 1

PFI-1

  • Target:

    Epigenetic Reader Domain|||Apoptosis|||Autophagy
  • Related Pathways:

    Chromatin/Epigenetic|||Apoptosis|||Autophagy
  • Purity:

    0.9919
  • Bioactivity:

    PFI-1 (PF-6405761), a specific BET (bromodomain-containing protein) inhibitor for BRD4, is with the IC50 of 0.22 ?M in a cell-free assay.
  • Smiles:

    COc1ccccc1S(=O)(=O)Nc1ccc2NC(=O)N(C)Cc2c1
  • Molecular Formula:

    C16H17N3O4S
  • Molecular Weight:

    347.39
  • Shipping Conditions:

    Cool pack
  • Storage Temperature:

    -20°C
  • CAS Number:

    1403764-72-6