Products for Research Use Only

PFI-2

CAT: 0931-T1987-01Size: 1 mgDry Ice: NoHazardous: No
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CAT#:0931-T1987-01Size:1 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
1627676-59-8
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9938
Bioactivity
PFI-2 is an effective, specific and cell-active lysine methyltransferase SETD7 inhibitor (Ki/IC50: 0.33/2 nM), 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.
Smiles
FC1=C2C(=CC(S(N[C@H](CC3=CC(C(F)(F)F)=CC=C3)C(=O)N4CCCC4)(=O)=O)=C1)CCNC2
Molecular Formula
C23H25F4N3O3S
Molecular Weight
499.52
Shipping Conditions
Ice Packs
Storage Temperature
-20°C