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MPT0G211 mesylate

CAT: 0931-T61753-01Size: 25 mgDry Ice: NoHazardous: No
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CAT#:0931-T61753-01Size:25 mg
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24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2151854-33-8
Target
Others, HDAC
Related Pathways
Others, DNA Damage/DNA Repair, Chromatin/Epigenetic
Bioactivity
MPT0G211 mesylate is a powerful and selective HDAC6 inhibitor (IC50 = 0.291 nM), with high oral bioavailability. It exhibits remarkable selectivity for HDAC6 over other HDAC isoforms (>1000-fold selectivity) . Additionally, MPT0G211 mesylate can effectively cross the blood-brain barrier. In preclinical studies using an Alzheimer's disease model, MPT0G211 mesylate has shown promising results in reducing tau phosphorylation and cognitive deficits. Furthermore, this compound exhibits anti-metastatic and neuroprotective effects, making it a potential candidate for anticancer interventions. [1] [2] [3].
Smiles
CS(O)(=O)=O.ONC(=O)c1ccc(CNc2cccc3cccnc23)cc1
Molecular Formula
C18H19N3O5S
Molecular Weight
389.43
Shipping Conditions
Ice Packs
Storage Temperature
-20°C

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