Tepotinib
- Availability: 24/48H Stock Items & 2 to 6 Weeks non Stock Items.
- Dry Ice Shipment: No


Tepotinib
Target:
C-Met/HGFR|||Autophagy|||TAM Receptor|||Trk receptorRelated Pathways:
Tyrosine Kinase/Adaptors|||AutophagyPurity:
0.9991Bioactivity:
Tepotinib (EMD-1214063) is a c-MET tyrosine kinase inhibitor (IC50=3 nM) that is selective, orally active, and ATP-competitive. Tepotinib has antitumor effect and is used in the treatment of non-small cell lung cancer.Smiles:
CN1CCC(COc2cnc(nc2)-c2cccc(Cn3nc(ccc3=O)-c3cccc(c3)C#N)c2)CC1Molecular Formula:
C29H28N6O2Molecular Weight:
492.57Shipping Conditions:
Cool packStorage Temperature:
-20°CCAS Number:
1100598-32-0
