GSK343

• Target:

  Histone Methyltransferase|||Autophagy

• Related Pathways:

  Autophagy|||Chromatin/Epigenetic

• Purity:

  0.999

• Bioactivity:

  GSK343, a specific and effective EZH2 inhibitor (IC50=4 nM), exhibits 60 fold specificity activity against EZH1, and >1000 fold specificity activity against other histone methyltransferases.

• Smiles:

  CCCc1cc(C)[nH]c(=O)c1CNC(=O)c1cc(cc2n(ncc12)C(C)C)-c1ccnc(c1)N1CCN(C)CC1

• Molecular Formula:

  C31H39N7O2

• Molecular Weight:

  541.69

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  1346704-33-3