PCSK9 modulator-2

• Target :

  Others

• Related Pathways :

  Others

• Bioactivity :

  PCSK9 modulator-2 (Compound 1) is a potent PCSK9 modulator (EC 50 = 202 nM) with potential applications in hyperlipidemia research. Proprotein convertase subtilisin/kexin type 9 (PCSK9) is a recently validated therapeutic target for lowering low-density lipoprotein cholesterol (LDL-C) [1].

• Smiles :

  C(C=1C=2C(NC1)=C(F)C=CC2)C=3NC=4C(C3)=CC(F)=CC4

• Molecular Formula :

  C17H12F2N2

• Molecular Weight :

  282.29

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2365416-53-9