PCSK9-IN-2

• Target :

  Others

• Related Pathways :

  Others

• Bioactivity :

  PCSK9-IN-2 is a newly developed small molecule that effectively inhibits the protein-protein interaction (PPI) between PCSK9 and LDLR. It has been found to have a potent inhibitory activity with an IC50 value of 7.57 ?M.

• Smiles :

  O=C1C[C@@H](N[C@@H]2CCCCNC2=O)C(=O)N1c1ccc(cc1)N1C(=O)C[C@@H](N[C@@H]2CCCCNC2=O)C1=O

• Molecular Formula :

  C26H32N6O6

• Molecular Weight :

  524.578

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C

• CAS Number :

  2099167-44-7