PF 429242

• CAS Number :

  947303-87-9

• Target :

  Fatty Acid Synthase|||Lipid|||Virus Protease|||NPC1L1

• Related Pathways :

  Microbiology/Virology|||Metabolism|||Membrane transporter/Ion channel

• Purity :

  0.9927

• Bioactivity :

  PF-429242 is a competitive inhibitor of sterol regulatory element-binding protein (SREBP) site 1 protease (IC50 = 0.175 ?M) . It is selective for site 1 protease against a panel of serine proteases. PF-429242 inhibits rate of cholesterol synthesis in CHO cells (IC50 = 0.53 ?M) .

• Smiles :

  N(C(=O)C1=CC=C(CN(CC)CC)C=C1)(CCC2=C(OC)C=CC=C2)[C@@H]3CCNC3

• Molecular Formula :

  C25H35N3O2

• Molecular Weight :

  409.56

• Shipping Conditions :

  Cool pack

• Storage Temperature :

  -20°C