Helianorphin-19

CAT: 0931-MF-0037503Size: 1 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0037503Size:1 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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Target
Opioid Receptor
Related Pathways
Neuroscience|||GPCR/G Protein|||Endocrinology/Hormones
Bioactivity
Helianorphin-19 is a high affinity, potent and selective ?-opioid receptor (KOR) agonist (Ki = 25 nM; EC50= 45 nM) . Helianorphin-19 exhibits approximately 200-fold selectivity for KOR over ? and ?-opioid receptors.In vivoHelianorphin-19 shows potent peripheral analgesic efficacy in a mouse model of visceral pain without affecting motor coordination/sedation.
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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