Products for Research Use Only

Helianorphin-19

CAT: 0931-T41183Size: 1 mgDry Ice: NoHazardous: No
Product image 1
1 / 1
CAT#:0931-T41183Size:1 mg
Selected
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
Quick Request Actions
Target
Opioid Receptor
Related Pathways
Neuroscience, GPCR/G Protein, Endocrinology/Hormones
Bioactivity
Helianorphin-19 is a high affinity, potent and selective κ-opioid receptor (KOR) agonist (Ki = 25 nM; EC50= 45 nM) . Helianorphin-19 exhibits approximately 200-fold selectivity for KOR over μ and δ-opioid receptors.In vivoHelianorphin-19 shows potent peripheral analgesic efficacy in a mouse model of visceral pain without affecting motor coordination/sedation.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C