EPZ-719

CAT: 0931-MF-0109868-01Size: 5 mgDry Ice: NoHazardous: No
CAT#:0931-MF-0109868-01Size:5 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
2697176-16-0
Target
Histone Methyltransferase|||Others
Related Pathways
Chromatin/Epigenetic|||Others
Bioactivity
EPZ-719 is a highly selective and potent inhibitor of SETD2, a novel compound known for its ability to inhibit the enzymatic activity of SETD2 (IC50 = 0.005 ?M) . This compound displays a remarkable selectivity over other histone methyltransferases, making it a promising candidate for targeted therapeutic applications in the field of epigenetic research.
Smiles
CN([C@H]1CCN(C1)[C@H]1CCC[C@H](C1)NC(=O)c1cc2c(F)ccc(C)c2[nH]1)S(C)(=O)=O
Molecular Formula
C22H31FN4O3S
Molecular Weight
450.57
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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