M-808

• Target:

  Others|||Epigenetic Reader Domain

• Related Pathways:

  Chromatin/Epigenetic|||Others

• Bioactivity:

  M-808 is a potent and efficacious covalent inhibitor, targeting the interaction between Menin and MLL. It demonstrates a high binding affinity with an IC50 value of 2.6 nM.

• Smiles:

  [H][C@@]1 (CCC[C@@H]1NC (=O) OC) [C@@] (CN1CCC1) (C1CCN (CC2CN (C2) c2ccc (cc2) S (=O) (=O) C2CN (C2) C (=O) \C=C\CN2CCCCC2) CC1) c1cccc (F) c1

• Molecular Formula:

  C45H63FN6O5S

• Molecular Weight:

  819.09

• Shipping Conditions:

  Cool pack

• Storage Temperature:

  -20°C

• CAS Number:

  2377335-74-3