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CAY10568

CAT: 0931-T37670-01Size: 10 mgDry Ice: NoHazardous: No
CAT#:0931-T37670-01Size:10 mg
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AVAILABILITY: InStock
24/48H Stock Items & 2 to 6 Weeks non Stock Items.
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CAS Number
22913-17-3
Target
Sodium Channel|||Others
Related Pathways
Others|||Membrane transporter/Ion channel
Bioactivity
Most local anesthetics act by abolishing voltage gated sodium channel currents indiscriminately in all populations of neurons. Selective analgesia through TRPV1-mediated entry of a cationic lidocaine derivative, QX314, was recently reported. CAY10568 is a physically smaller, less hydrophobic version of QX314 designed to be even more permeable to TRPV1 ion channel when activated by agonists such as capsaicin and N-oleoyl dopamine. CAY10568 when given in combination with suitable TRPV1 agonists should produce selective blockade of the pain response while leaving motor, touch, and proprioception intact.
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[I-].C[N+](C)(C)CC(=O)Nc1ccccc1
Molecular Formula
C11H17IN2O
Molecular Weight
320.174
Shipping Conditions
Cool pack
Storage Temperature
-20°C

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